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159093 (1S)-(αR,3aS,4S,6S,7aR)-Hexahydro-3a,8,8-trimethyl-α-pentyl-4,6-methano-1,3,2-benzodioxaborole-2-methanamine Trifluoroacetic Acid Salt CAS:

Specifications

References

Grade

Highly Purified

Molecular Formula

C18H31BF3NO4

Molecular Weight

393.25

EU Commodity Code

38220090

Shipping Temp

Blue Ice

Storage Temp

-20°C

(αR,3aS,4S,6S,7aR)-Hexahydro-3a,5,5-trimethyl-α-pentyl-4,6-methano-1,3,2-benzodioxaborole-2-methanamine Trifluoroacetic Acid Salt

(αR,3aS,4S,6S,7aR)-Hexahydro-3a,8,8-trimethyl-α-pentyl-4,6-methano-1,3,2-benzodioxaborole-2-methanamine is an intermediate in the preparation of Bortezomib (B675700), a dipeptidyl boronate proteasome inhibitor.

Solubility

Acetone, Ethyl Acetate

References

Zhu, Y., et al.: Bioorg. Med. Chem., 14, 1483 (2006), �Dorsey, B., et al.: J. Med. Chem., 51, 1068 (2008), Zhu, Y., et al.: Eur. J .Med. Chem., 44, 1486� (2009),