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007087 CP-154526 Hydrochloride CAS: 257639-98-8

Specifications
References
CAS Number
257639-98-8
Grade
Highly Purified
Molecular Formula
C23H33ClN4
Molecular Weight
400.99
EU Commodity Code
38220090
Shipping Temp
RT
Storage Temp
4°C
N-Butyl-N-ethyl-2,5-dimethyl-7-(2,4,6-trimethylphenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine Hydrochloride

A selective, non-peptide antagonist of corticotropin releasing factor receptors (CRF1). It blocks CRF-induced adenylate cyclase activation and attenuates activation of the HPA axis by CRF. It displayed anxiolytic-like activity in the rat elevated plus-maze test; brain penetrant.

Form
Pale Yellow Solid
Melting Point
167-169°C
Solubility
DMSO, Methanol
Pfizer Compound
References
Lundkist, J. et al.: Eur. J. Pharmacol., 309, 195 (1996); Arbolius, L. et al.: J. pharmacol. Exp. Therap., 294, 588 (2000); Kehne, J.H. et al.: Neuropharmacol., 39, 1357 (2000);
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